GPCR focused libraries - new products from OTAVA

Otava releases two GPCR-related focused libraries. The libraries have been designed with QSAR using training set. These libraries are proposed for screening in GPCR-associated research and drug development.
By: Andrey Grischenko
 
Oct. 2, 2009 - PRLog -- We are happy to offer Otava’s  two GPCR-related focused libraries:

1. GPCR Antagonist focused library (4953 compounds)
2. GPCR Agonists focused library (466 compounds)

The libraries have been designed with QSAR using training set of compounds active towards various GPCRs .  The libraries contain drug-like compounds having the following predicted activities:

GPCR Antagonist focused library   
5 Hydroxytryptamine antagonist   
Acetylcholine muscarinic antagonist   
Adenosine receptor antagonist   
Alpha adrenoreceptor antagonist   
Beta adrenoreceptor antagonist   
Endothelin receptor antagonist
GABA receptor antagonist
Dopamine antagonist   
Glucagon receptor antagonist   
Glutamate receptor antagonist   
Histamine antagonist   
Melatonin antagonist   
Neuropeptide antagonist   
Prostaglandin antagonist   
Thromboxane antagonist   
Vasopressin 1 antagonist

GPCR Agonist focused library   
5 Hydroxytryptamine agonist
Acetylcholine muscarinic agonist
Alpha adrenoreceptor agonist
Beta adrenoreceptor agonist
Cholecystokinin agonist
Dopamine agonist
Dopamine autoreceptor agonist
GABA receptor agonist
Melatonin agonist


All compounds are in stock, cherry-picking is available.  These libraries are proposed for screening in GPCR-associated research and drug development.
End
Source:Andrey Grischenko
Email:***@otavachemicals.com
Zip:03143
Tags:Gpcr, Focused Library
Industry:Biotech
Location:Kyiv - Kyiv - Ukraine
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